| Title | Date | PubMed ID |
|---|
| Characterization of DprE1-Mediated Benzothiazinone Resistance in Mycobacterium tuberculosis. | 2016 Nov | 27527085 |
| Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure-activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-D-ribose 2'-oxidase. | 2015 Dec 15 | 26643218 |
| Whole Cell Target Engagement Identifies Novel Inhibitors of Mycobacterium tuberculosis Decaprenylphosphoryl-β-d-ribose Oxidase. | 2015 Dec 11 | 27623058 |
| The 8-Pyrrole-Benzothiazinones Are Noncovalent Inhibitors of DprE1 from Mycobacterium tuberculosis. | 2015 Aug | 25987616 |
| Structure, dynamics, and interaction of Mycobacterium tuberculosis (Mtb) DprE1 and DprE2 examined by molecular modeling, simulation, and electrostatic studies. | 2015 | 25789990 |
| 4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity. | 2014 Jun 26 | 24871036 |
| Discovery of pyrazolopyridones as a novel class of noncovalent DprE1 inhibitor with potent anti-mycobacterial activity. | 2014 Jun 12 | 24818517 |
| The DprE1 enzyme, one of the most vulnerable targets of Mycobacterium tuberculosis. | 2013 Oct | 24037308 |
| Crystal structure of decaprenylphosphoryl-β- D-ribose 2'-epimerase from Mycobacterium smegmatis. | 2013 Mar | 23184707 |
| Structural basis of inhibition of Mycobacterium tuberculosis DprE1 by benzothiazinone inhibitors. | 2012 Jul 10 | 22733761 |