TitleDatePubMed ID
Pharmacophore mapping, molecular docking, chemical synthesis of some novel pyrrolyl benzamide derivatives and evaluation of their inhibitory activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis.2018 Dec30223149
Discovery of a cofactor-independent inhibitor of <i>Mycobacterium tuberculosis</i> InhA.2018 Jun30456352
An overview on crystal structures of InhA protein: Apo-form, in complex with its natural ligands and inhibitors.2018 Feb 2529407960
Evaluating the Contribution of Transition-State Destabilization to Changes in the Residence Time of Triazole-Based InhA Inhibitors.2017 Mar 828151657
N-Benzyl-4-((heteroaryl)methyl)benzamides: A New Class of Direct NADH-Dependent 2-trans Enoyl-Acyl Carrier Protein Reductase (InhA) Inhibitors with Antitubercular Activity.2016 Apr 526934341
Piperazine derivatives: synthesis, inhibition of the Mycobacterium tuberculosis enoyl-acyl carrier protein reductase and SAR studies.2015 Jan 2725461892
Development of 2-(4-oxoquinazolin-3(4H)-yl)acetamide derivatives as novel enoyl-acyl carrier protein reductase (InhA) inhibitors for the treatment of tuberculosis.2014 Oct 3025218910
Conformational changes in 2-trans-enoyl-ACP (CoA) reductase (InhA) from M. tuberculosis induced by an inorganic complex: a molecular dynamics simulation study.2012 May21833828
Targeting InhA, the FASII enoyl-ACP reductase: SAR studies on novel inhibitor scaffolds.201222283812
Phosphorylation of InhA inhibits mycolic acid biosynthesis and growth of Mycobacterium tuberculosis.2010 Dec21143326