Substance-K receptor
Name | Substance-K receptor |
---|---|
Synonyms | Neurokinin A receptor NK-2 receptor NK-2R NK2R NKNAR SKR TAC2R Tachykinin receptor 2 |
Gene Name | TACR2 |
Organism | Human |
Amino acid sequence | >lcl|BSEQ0016718|Substance-K receptor MGTCDIVTEANISSGPESNTTGITAFSMPSWQLALWATAYLALVLVAVTGNAIVIWIILA HRRMRTVTNYFIVNLALADLCMAAFNAAFNFVYASHNIWYFGRAFCYFQNLFPITAMFVS IYSMTAIAADRYMAIVHPFQPRLSAPSTKAVIAGIWLVALALASPQCFYSTVTMDQGATK CVVAWPEDSGGKTLLLYHLVVIALIYFLPLAVMFVAYSVIGLTLWRRAVPGHQAHGANLR HLQAMKKFVKTMVLVVLTFAICWLPYHLYFILGSFQEDIYCHKFIQQVYLALFWLAMSST MYNPIIYCCLNHRFRSGFRLAFRCCPWVTPTKEDKLELTPTTSLSTRVNRCHTKETLFMA GDTAPSEATSGEAGRPQDGSGLWFGYGLLAPTKTHVEI |
Number of residues | 398 |
Molecular Weight | 44441.705 |
Theoretical pI | 8.74 |
GO Classification |
Functions
tachykinin receptor activity substance K receptor activity Processes
response to electrical stimulus tachykinin receptor signaling pathway muscle contraction prolactin secretion intestine smooth muscle contraction neuropeptide signaling pathway positive regulation of uterine smooth muscle contraction synaptic transmission operant conditioning positive regulation of vascular permeability positive regulation of smooth muscle contraction positive regulation of acetylcholine secretion, neurotransmission cell surface receptor signaling pathway negative regulation of luteinizing hormone secretion excretion Components
plasma membrane integral component of plasma membrane |
General Function | Tachykinin receptor activity |
Specific Function | This is a receptor for the tachykinin neuropeptide substance K (neurokinin A). It is associated with G proteins that activate a phosphatidylinositol-calcium second messenger system. The rank order of affinity of this receptor to tachykinins is: substance K > neuromedin-K > substance P. |
Transmembrane Regions | 33-56 70-90 108-129 150-170 197-218 252-272 291-310 |
GenBank Protein ID | 189135 |
UniProtKB ID | P21452 |
UniProtKB Entry Name | NK2R_HUMAN |
Cellular Location | Cell membrane |
Gene sequence | >lcl|BSEQ0016719|Substance-K receptor (TACR2) ATGGGGACCTGTGACATTGTGACTGAAGCCAATATCTCATCTGGCCCTGAGAGCAACACC ACGGGCATCACAGCCTTCTCCATGCCCAGCTGGCAACTGGCACTGTGGGCCACAGCCTAC CTGGCCCTGGTGCTGGTGGCCGTGACGGGTAATGCCATCGTCATCTGGATCATCCTGGCC CATCGGAGGATGCGCACAGTCACCAACTACTTCATCGTCAATCTGGCGCTGGCTGACCTC TGCATGGCTGCCTTCAATGCCGCCTTCAACTTTGTCTATGCCAGCCACAACATCTGGTAC TTTGGCCGTGCCTTCTGCTACTTCCAGAACCTCTTCCCCATCACAGCCATGTTTGTCAGC ATCTACTCCATGACCGCCATTGCTGCCGACAGGTACATGGCCATCGTCCACCCCTTCCAG CCTCGGCTTTCAGCTCCCAGCACCAAGGCGGTTATTGCTGGCATCTGGCTGGTGGCTCTC GCCCTGGCCTCCCCTCAGTGCTTCTACTCCACCGTCACCATGGACCAGGGTGCCACCAAG TGCGTGGTGGCCTGGCCCGAAGACAGCGGGGGCAAGACGCTCCTCCTGTACCACCTCGTG GTGATCGCCCTCATCTACTTCCTGCCGCTCGCGGTGATGTTTGTAGCCTACAGCGTCATC GGCCTCACGCTCTGGAGGCGCGCAGTGCCCGGACATCAGGCGCACGGTGCCAACCTGCGC CACCTGCAGGCCATGAAGAAGTTTGTGAAGACCATGGTGCTGGTGGTGCTGACGTTTGCC ATCTGCTGGCTGCCCTACCACCTCTACTTCATCCTGGGCAGCTTCCAGGAGGACATCTAC TGCCACAAGTTCATCCAGCAAGTCTACCTGGCACTCTTCTGGTTGGCCATGAGCTCTACC ATGTACAATCCCATCATCTACTGCTGTCTCAACCACAGGTTTCGCTCTGGATTCCGGCTT GCCTTCCGCTGCTGCCCATGGGTCACACCCACCAAGGAAGATAAGCTCGAGCTGACTCCC ACGACCTCCCTCTCCACGAGAGTCAACAGGTGTCACACTAAGGAGACTTTGTTCATGGCT GGGGACACAGCCCCCTCCGAGGCTACCAGTGGGGAGGCGGGGCGTCCCCAGGATGGATCA GGGCTATGGTTTGGGTATGGTTTGCTTGCCCCCACCAAAACTCATGTTGAAATTTGA |
GenBank Gene ID | M57414 |
GeneCard ID | None |
GenAtlas ID | TACR2 |
HGNC ID | HGNC:11527 |
Chromosome Location | 10 |
Locus | 10q11-q21 |
References |
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Related FRC
FRCD ID | Name | Exact Mass | Structure |
---|---|---|---|
Captan |
300.578 |
||
Fenhexamid |
302.195 |
||
Mercuric chloride |
271.492 |