P2X purinoceptor 4
Name | P2X purinoceptor 4 |
---|---|
Synonyms | ATP receptor P2X4 Purinergic receptor |
Gene Name | P2RX4 |
Organism | Human |
Amino acid sequence | >lcl|BSEQ0009820|P2X purinoceptor 4 MAGCCAALAAFLFEYDTPRIVLIRSRKVGLMNRAVQLLILAYVIGWVFVWEKGYQETDSV VSSVTTKVKGVAVTNTSKLGFRIWDVADYVIPAQEENSLFVMTNVILTMNQTQGLCPEIP DATTVCKSDASCTAGSAGTHSNGVSTGRCVAFNGSVKTCEVAAWCPVEDDTHVPQPAFLK AAENFTLLVKNNIWYPKFNFSKRNILPNITTTYLKSCIYDAKTDPFCPIFRLGKIVENAG HSFQDMAVEGGIMGIQVNWDCNLDRAASLCLPRYSFRRLDTRDVEHNVSPGYNFRFAKYY RDLAGNEQRTLIKAYGIRFDIIVFGKAGKFDIIPTMINIGSGLALLGMATVLCDIIVLYC MKKRLYYREKKYKYVEDYEQGLASELDQ |
Number of residues | 388 |
Molecular Weight | 43368.725 |
Theoretical pI | None |
GO Classification |
Functions
ATP binding copper ion binding receptor binding cadherin binding drug binding protein homodimerization activity zinc ion binding extracellular ATP-gated cation channel activity purinergic nucleotide receptor activity Processes
signal transduction nitric oxide biosynthetic process ion transmembrane transport endothelial cell activation regulation of cardiac muscle contraction negative regulation of cardiac muscle hypertrophy regulation of blood pressure positive regulation of nitric oxide biosynthetic process sensory perception of pain apoptotic signaling pathway positive regulation of calcium ion transport cellular response to ATP protein homooligomerization relaxation of cardiac muscle vasodilation positive regulation of calcium ion transport into cytosol membrane depolarization transport excitatory postsynaptic potential neuronal action potential regulation of sodium ion transport response to fluid shear stress calcium ion transport response to ATP tissue homeostasis positive regulation of prostaglandin secretion positive regulation of calcium-mediated signaling purinergic nucleotide receptor signaling pathway Components
neuronal cell body apical part of cell postsynaptic density plasma membrane dendritic spine cell junction lysosomal membrane terminal bouton extracellular exosome integral component of nuclear inner membrane perinuclear region of cytoplasm integral component of plasma membrane membrane |
General Function | Zinc ion binding |
Specific Function | Receptor for ATP that acts as a ligand-gated ion channel. This receptor is insensitive to the antagonists PPADS and suramin. |
Transmembrane Regions | 34-54 339-359 |
GenBank Protein ID | |
UniProtKB ID | Q99571 |
UniProtKB Entry Name | P2RX4_HUMAN |
Cellular Location | Membrane |
Gene sequence | >lcl|BSEQ0013934|P2X purinoceptor 4 (P2RX4) ATGGCGGGCTGCTGCGCCGCGCTGGCGGCCTTCCTGTTCGAGTACGACACGCCGCGCATC GTGCTCATCCGCAGCCGCAAAGTGGGGCTCATGAACCGCGCCGTGCAACTGCTCATCCTG GCCTACGTCATCGGGTGCTACCATCCCCATTTGGCAGAAGTGGAAATGGAGTCCCCTAGA AGGTGGGTGTTTGTGTGGGAAAAGGGCTACCAGGAAACTGACTCCGTGGTCAGCTCCGTT ACGACCAAGGTCAAGGGCGTGGCTGTGACCAACACTTCTAAACTTGGATTCCGGATCTGG GATGTGGCGGATTATGTGATACCAGCTCAGGAGGAAAACTCCCTCTTCGTCATGACCAAC GTGATCCTCACCATGAACCAGACACAGGGCCTGTGCCCCGAGATTCCAGATGCGACCACT GTGTGTAAATCAGATGCCAGCTGTACTGCCGGCTCTGCCGGCACCCACAGCAACGGAGTC TCAACAGGCAGGTGCGTAGCTTTCAACGGGTCTGTCAAGACGTGTGAGGTGGCGGCCTGG TGCCCGGTGGAGGATGACACACACGTGCCACAACCTGCTTTTTTAAAGGCTGCAGAAAAC TTCACTCTTTTGGTTAAGAACAACATCTGGTATCCCAAATTTAATTTCAGCAAGAGGAAT ATCCTTCCCAACATCACCACTACTTACCTCAAGTCGTGCATTTATGATGCTAAAACAGAT CCCTTCTGCCCCATATTCCGTCTTGGCAAAATAGTGGAGAACGCAGGACACAGTTTCCAG GACATGGCCGTGGAGGGAGGCATCATGGGCATCCAGGTCAACTGGGACTGCAACCTGGAC AGAGCCGCCTCCCTCTGCTTGCCCAGGTACTCCTTCCGCCGCCTCGATACACGGGACGTT GAGCACAACGTATCTCCTGGCTACAATTTCAGGTTTGCCAAGTACTACAGAGACCTGGCT GGCAACGAGCAGCGCACGCTCATCAAGGCCTATGGCATCCGCTTCGACATCATTGTGTTT GGGAAGGCAGGGAAATTTGACATCATCCCCACTATGATCAACATCGGCTCTGGCCTGGCA CTGCTAGGCATGGCGACCGTGCTGTGTGACATCATAGTCCTCTACTGCATGAAGAAAAGA CTCTACTATCGGGAGAAGAAATATAAATATGTGGAAGATTACGAGCAGGGTCTTGCTAGT GAGCTGGACCAGTGA |
GenBank Gene ID | |
GeneCard ID | None |
GenAtlas ID | |
HGNC ID | HGNC:8535 |
Chromosome Location | 12 |
Locus | None |
References |
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Related FRC
FRCD ID | Name | Exact Mass | Structure |
---|---|---|---|
Paroxetine |
329.4 |