Histamine H4 receptor
Name | Histamine H4 receptor |
---|---|
Synonyms | AXOR35 G-protein coupled receptor 105 GPCR105 GPRv53 H4R Pfi-013 SP9144 |
Gene Name | HRH4 |
Organism | Human |
Amino acid sequence | >lcl|BSEQ0000291|Histamine H4 receptor MPDTNSTINLSLSTRVTLAFFMSLVAFAIMLGNALVILAFVVDKNLRHRSSYFFLNLAIS DFFVGVISIPLYIPHTLFEWDFGKEICVFWLTTDYLLCTASVYNIVLISYDRYLSVSNAV SYRTQHTGVLKIVTLMVAVWVLAFLVNGPMILVSESWKDEGSECEPGFFSEWYILAITSF LEFVIPVILVAYFNMNIYWSLWKRDHLSRCQSHPGLTAVSSNICGHSFRGRLSSRRSLSA STEVPASFHSERQRRKSSLMFSSRTKMNSNTIASKMGSFSQSDSVALHQREHVELLRARR LAKSLAILLGVFAVCWAPYSLFTIVLSFYSSATGPKSVWYRIAFWLQWFNSFVNPLLYPL CHKRFQKAFLKIFCIKKQPLPSQHSRSVSS |
Number of residues | 390 |
Molecular Weight | 44495.375 |
Theoretical pI | 9.92 |
GO Classification |
Functions
histamine receptor activity histamine binding Processes
negative regulation of adenylate cyclase activity regulation of MAPK cascade inflammatory response positive regulation of cytosolic calcium ion concentration sensory perception of chemical stimulus Components
plasma membrane cytosol integral component of plasma membrane |
General Function | Histamine receptor activity |
Specific Function | The H4 subclass of histamine receptors could mediate the histamine signals in peripheral tissues. Displays a significant level of constitutive activity (spontaneous activity in the absence of agonist). |
Transmembrane Regions | 20-40 53-73 88-108 132-152 173-193 305-325 342-362 |
GenBank Protein ID | 10241847 |
UniProtKB ID | Q9H3N8 |
UniProtKB Entry Name | HRH4_HUMAN |
Cellular Location | Cell membrane |
Gene sequence | >lcl|BSEQ0009967|Histamine H4 receptor (HRH4) ATGCCAGATACTAATAGCACAATCAATTTATCACTAAGCACTCGTGTTACTTTAGCATTT TTTATGTCCTTAGTAGCTTTTGCTATAATGCTAGGAAATGCTTTGGTCATTTTAGCTTTT GTGGTGGACAAAAACCTTAGACATCGAAGTAGTTATTTTTTTCTTAACTTGGCCATCTCT GACTTCTTTGTGGTTTCAGAGTCTTGGAAGGATGAAGGTAGTGAATGTGAACCTGGATTT TTTTCGGAATGGTACATCCTTGCCATCACATCATTCTTGGAATTCGTGATCCCAGTCATC TTAGTCGCTTATTTCAACATGAATATTTATTGGAGCCTGTGGAAGCGTGATCATCTCAGT AGGTGCCAAAGCCATCCTGGACTGACTGCTGTCTCTTCCAACATCTGTGGACACTCATTC AGAGGTAGACTATCTTCAAGGAGATCTCTTTCTGCATCGACAGAAGTTCCTGCATCCTTT CATTCAGAGAGACAGAGGAGAAAGAGTAGTCTCATGTTTTCCTCAAGAACCAAGATGAAT AGCAATACAATTGCTTCCAAAATGGGTTCCTTCTCCCAATCAGATTCTGTAGCTCTTCAC CAAAGGGAACATGTTGAACTGCTTAGAGCCAGGAGATTAGCCAAGTCACTGGCCATTCTC TTAGGGGTTTTTGCTGTTTGCTGGGCTCCATATTCTCTGTTCACAATTGTCCTTTCATTT TATTCCTCAGCAACAGGTCCTAAATCAGTTTGGTATAGAATTGCATTTTGGCTTCAGTGG TTCAATTCCTTTGTCAATCCTCTTTTGTATCCATTGTGTCACAAGCGCTTTCAAAAGGCT TTCTTGAAAATATTTTGTATAAAAAAGCAACCTCTACCATCACAACACAGTCGGTCAGTA TCTTCTTAA |
GenBank Gene ID | AB044934 |
GeneCard ID | None |
GenAtlas ID | HRH4 |
HGNC ID | HGNC:17383 |
Chromosome Location | 18 |
Locus | 18q11.2 |
References |
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