Absorption |
Blood-Brain Barrier | BBB+ | 0.9080 |
Human Intestinal Absorption | HIA+ | 0.9333 |
Caco-2 Permeability | Caco2- | 0.6448 |
P-glycoprotein Substrate | Non-substrate | 0.8964 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9323 |
Non-inhibitor | 0.9954 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9442 |
Distribution |
Subcellular localization | Mitochondria | 0.4648 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8246 |
CYP450 2D6 Substrate | Non-substrate | 0.8284 |
CYP450 3A4 Substrate | Non-substrate | 0.7604 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8662 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8555 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9145 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8640 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9886 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9650 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.7724 |
Non-inhibitor | 0.9337 |
AMES Toxicity | Non AMES toxic | 0.8646 |
Carcinogens | Carcinogens | 0.8323 |
Fish Toxicity | Low FHMT | 0.7029 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7580 |
Honey Bee Toxicity | High HBT | 0.7693 |
Biodegradation | Ready biodegradable | 0.5873 |
Acute Oral Toxicity | III | 0.6748 |
Carcinogenicity (Three-class) | Non-required | 0.6637 |