Absorption |
Blood-Brain Barrier | BBB+ | 0.9742 |
Human Intestinal Absorption | HIA+ | 0.9502 |
Caco-2 Permeability | Caco2+ | 0.5968 |
P-glycoprotein Substrate | Non-substrate | 0.8714 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9900 |
Non-inhibitor | 0.9920 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9466 |
Distribution |
Subcellular localization | Mitochondria | 0.6597 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.7913 |
CYP450 2D6 Substrate | Non-substrate | 0.9384 |
CYP450 3A4 Substrate | Non-substrate | 0.7921 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8774 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9482 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9667 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9786 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9854 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9818 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9666 |
Non-inhibitor | 0.9889 |
AMES Toxicity | Non AMES toxic | 0.9635 |
Carcinogens | Carcinogens | 0.6222 |
Fish Toxicity | Low FHMT | 0.5188 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9789 |
Honey Bee Toxicity | High HBT | 0.7907 |
Biodegradation | Ready biodegradable | 0.9758 |
Acute Oral Toxicity | III | 0.7885 |
Carcinogenicity (Three-class) | Non-required | 0.6783 |