Absorption |
Blood-Brain Barrier | BBB+ | 0.6165 |
Human Intestinal Absorption | HIA+ | 0.9756 |
Caco-2 Permeability | Caco2+ | 0.8867 |
P-glycoprotein Substrate | Non-substrate | 0.7340 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9815 |
Non-inhibitor | 0.9937 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9167 |
Distribution |
Subcellular localization | Mitochondria | 0.8764 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.7962 |
CYP450 2D6 Substrate | Non-substrate | 0.9233 |
CYP450 3A4 Substrate | Non-substrate | 0.7660 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9517 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.7984 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9659 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.7644 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.8675 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.8525 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9631 |
Non-inhibitor | 0.9734 |
AMES Toxicity | Non AMES toxic | 0.9829 |
Carcinogens | Non-carcinogens | 0.8627 |
Fish Toxicity | High FHMT | 0.7460 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7307 |
Honey Bee Toxicity | High HBT | 0.7317 |
Biodegradation | Ready biodegradable | 0.8086 |
Acute Oral Toxicity | III | 0.7939 |
Carcinogenicity (Three-class) | Non-required | 0.7871 |