Absorption |
Blood-Brain Barrier | BBB+ | 0.9639 |
Human Intestinal Absorption | HIA+ | 0.9841 |
Caco-2 Permeability | Caco2+ | 0.5644 |
P-glycoprotein Substrate | Non-substrate | 0.8563 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9888 |
Non-inhibitor | 0.9904 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9472 |
Distribution |
Subcellular localization | Mitochondria | 0.6703 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.7598 |
CYP450 2D6 Substrate | Non-substrate | 0.9517 |
CYP450 3A4 Substrate | Non-substrate | 0.8093 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9406 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9695 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9729 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9907 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9827 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9930 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9770 |
Non-inhibitor | 0.9876 |
AMES Toxicity | Non AMES toxic | 0.9815 |
Carcinogens | Carcinogens | 0.6452 |
Fish Toxicity | Low FHMT | 0.6462 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9428 |
Honey Bee Toxicity | High HBT | 0.7866 |
Biodegradation | Ready biodegradable | 0.9069 |
Acute Oral Toxicity | III | 0.7890 |
Carcinogenicity (Three-class) | Non-required | 0.7376 |