Absorption |
Blood-Brain Barrier | BBB+ | 0.9623 |
Human Intestinal Absorption | HIA+ | 0.7159 |
Caco-2 Permeability | Caco2- | 0.6276 |
P-glycoprotein Substrate | Non-substrate | 0.9043 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9006 |
Non-inhibitor | 0.9860 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9549 |
Distribution |
Subcellular localization | Mitochondria | 0.4783 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8506 |
CYP450 2D6 Substrate | Non-substrate | 0.8149 |
CYP450 3A4 Substrate | Non-substrate | 0.6946 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.7127 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.6684 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9057 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.6794 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9782 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9412 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9280 |
Non-inhibitor | 0.9362 |
AMES Toxicity | AMES toxic | 0.5087 |
Carcinogens | Carcinogens | 0.7796 |
Fish Toxicity | Low FHMT | 0.5324 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7816 |
Honey Bee Toxicity | High HBT | 0.8007 |
Biodegradation | Ready biodegradable | 0.9812 |
Acute Oral Toxicity | III | 0.6143 |
Carcinogenicity (Three-class) | Non-required | 0.6653 |