Absorption |
Blood-Brain Barrier | BBB+ | 0.8487 |
Human Intestinal Absorption | HIA+ | 0.9812 |
Caco-2 Permeability | Caco2- | 0.5452 |
P-glycoprotein Substrate | Non-substrate | 0.7597 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9752 |
Non-inhibitor | 0.9870 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9642 |
Distribution |
Subcellular localization | Mitochondria | 0.5364 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8116 |
CYP450 2D6 Substrate | Non-substrate | 0.9000 |
CYP450 3A4 Substrate | Non-substrate | 0.8100 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9244 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9434 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9679 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9741 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9297 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9736 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9623 |
Non-inhibitor | 0.9689 |
AMES Toxicity | Non AMES toxic | 0.9426 |
Carcinogens | Carcinogens | 0.5941 |
Fish Toxicity | Low FHMT | 0.5475 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9567 |
Honey Bee Toxicity | High HBT | 0.6091 |
Biodegradation | Ready biodegradable | 0.9434 |
Acute Oral Toxicity | III | 0.8497 |
Carcinogenicity (Three-class) | Non-required | 0.6947 |