Absorption |
Blood-Brain Barrier | BBB+ | 0.9692 |
Human Intestinal Absorption | HIA+ | 0.9937 |
Caco-2 Permeability | Caco2+ | 0.7277 |
P-glycoprotein Substrate | Non-substrate | 0.8235 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9639 |
Non-inhibitor | 0.9156 |
Renal Organic Cation Transporter | Non-inhibitor | 0.8964 |
Distribution |
Subcellular localization | Lysosome | 0.5206 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.7325 |
CYP450 2D6 Substrate | Non-substrate | 0.9212 |
CYP450 3A4 Substrate | Non-substrate | 0.7860 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.7394 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9447 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9708 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9088 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9638 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.8806 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.8975 |
Non-inhibitor | 0.9709 |
AMES Toxicity | Non AMES toxic | 0.6431 |
Carcinogens | Carcinogens | 0.7110 |
Fish Toxicity | Low FHMT | 0.5917 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9787 |
Honey Bee Toxicity | High HBT | 0.8239 |
Biodegradation | Ready biodegradable | 0.7450 |
Acute Oral Toxicity | III | 0.7858 |
Carcinogenicity (Three-class) | Non-required | 0.6287 |