Absorption |
Blood-Brain Barrier | BBB+ | 0.9623 |
Human Intestinal Absorption | HIA+ | 1.0000 |
Caco-2 Permeability | Caco2+ | 0.5499 |
P-glycoprotein Substrate | Non-substrate | 0.9016 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9371 |
Non-inhibitor | 0.9912 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9160 |
Distribution |
Subcellular localization | Mitochondria | 0.5613 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8679 |
CYP450 2D6 Substrate | Non-substrate | 0.8801 |
CYP450 3A4 Substrate | Non-substrate | 0.7173 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.7189 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9289 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.8908 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8499 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9831 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9125 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.7834 |
Non-inhibitor | 0.9729 |
AMES Toxicity | AMES toxic | 0.6901 |
Carcinogens | Carcinogens | 0.7654 |
Fish Toxicity | Low FHMT | 0.9178 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.5812 |
Honey Bee Toxicity | High HBT | 0.7743 |
Biodegradation | Ready biodegradable | 0.9541 |
Acute Oral Toxicity | II | 0.6926 |
Carcinogenicity (Three-class) | Warning | 0.4606 |