Absorption |
Blood-Brain Barrier | BBB+ | 0.9821 |
Human Intestinal Absorption | HIA+ | 0.9532 |
Caco-2 Permeability | Caco2+ | 0.7894 |
P-glycoprotein Substrate | Non-substrate | 0.7278 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9737 |
Non-inhibitor | 0.9794 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9278 |
Distribution |
Subcellular localization | Plasma membrane | 0.5164 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8124 |
CYP450 2D6 Substrate | Non-substrate | 0.8920 |
CYP450 3A4 Substrate | Non-substrate | 0.7109 |
CYP450 1A2 Inhibitor | Inhibitor | 0.6447 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9160 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9387 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9335 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9778 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9408 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9007 |
Non-inhibitor | 0.9234 |
AMES Toxicity | Non AMES toxic | 0.9863 |
Carcinogens | Carcinogens | 0.5208 |
Fish Toxicity | High FHMT | 0.8058 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7478 |
Honey Bee Toxicity | High HBT | 0.6796 |
Biodegradation | Ready biodegradable | 0.9752 |
Acute Oral Toxicity | III | 0.8736 |
Carcinogenicity (Three-class) | Non-required | 0.6618 |