Absorption |
Blood-Brain Barrier | BBB+ | 0.9733 |
Human Intestinal Absorption | HIA+ | 0.9601 |
Caco-2 Permeability | Caco2+ | 0.7678 |
P-glycoprotein Substrate | Non-substrate | 0.7508 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9694 |
Non-inhibitor | 0.9529 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9165 |
Distribution |
Subcellular localization | Plasma membrane | 0.5815 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8259 |
CYP450 2D6 Substrate | Non-substrate | 0.8816 |
CYP450 3A4 Substrate | Non-substrate | 0.7086 |
CYP450 1A2 Inhibitor | Inhibitor | 0.6209 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8936 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9367 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9283 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9709 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9424 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.8596 |
Non-inhibitor | 0.9129 |
AMES Toxicity | Non AMES toxic | 0.9785 |
Carcinogens | Non-carcinogens | 0.5055 |
Fish Toxicity | High FHMT | 0.9205 |
Tetrahymena Pyriformis Toxicity | High TPT | 0.8930 |
Honey Bee Toxicity | High HBT | 0.6747 |
Biodegradation | Ready biodegradable | 0.9697 |
Acute Oral Toxicity | III | 0.7683 |
Carcinogenicity (Three-class) | Non-required | 0.6955 |