Absorption |
Blood-Brain Barrier | BBB+ | 0.6903 |
Human Intestinal Absorption | HIA+ | 0.7413 |
Caco-2 Permeability | Caco2- | 0.7476 |
P-glycoprotein Substrate | Non-substrate | 0.5306 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9533 |
Non-inhibitor | 0.9220 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9414 |
Distribution |
Subcellular localization | Mitochondria | 0.8615 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8213 |
CYP450 2D6 Substrate | Non-substrate | 0.8714 |
CYP450 3A4 Substrate | Non-substrate | 0.6596 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8313 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8993 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9532 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9256 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9227 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9876 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9710 |
Non-inhibitor | 0.8664 |
AMES Toxicity | Non AMES toxic | 0.9468 |
Carcinogens | Non-carcinogens | 0.8642 |
Fish Toxicity | High FHMT | 0.6212 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8395 |
Honey Bee Toxicity | High HBT | 0.5275 |
Biodegradation | Ready biodegradable | 0.9863 |
Acute Oral Toxicity | III | 0.4938 |
Carcinogenicity (Three-class) | Non-required | 0.7834 |