Absorption |
Blood-Brain Barrier | BBB+ | 0.9647 |
Human Intestinal Absorption | HIA+ | 0.7887 |
Caco-2 Permeability | Caco2- | 0.5173 |
P-glycoprotein Substrate | Non-substrate | 0.8606 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9810 |
Non-inhibitor | 0.9857 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9554 |
Distribution |
Subcellular localization | Mitochondria | 0.7655 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8341 |
CYP450 2D6 Substrate | Non-substrate | 0.9298 |
CYP450 3A4 Substrate | Non-substrate | 0.7844 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9137 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9264 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9486 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9485 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9524 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9770 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9714 |
Non-inhibitor | 0.9929 |
AMES Toxicity | Non AMES toxic | 0.7926 |
Carcinogens | Non-carcinogens | 0.5114 |
Fish Toxicity | High FHMT | 0.9000 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9427 |
Honey Bee Toxicity | High HBT | 0.7806 |
Biodegradation | Ready biodegradable | 0.9713 |
Acute Oral Toxicity | III | 0.6058 |
Carcinogenicity (Three-class) | Non-required | 0.6842 |