Absorption |
Blood-Brain Barrier | BBB+ | 0.7144 |
Human Intestinal Absorption | HIA+ | 0.9418 |
Caco-2 Permeability | Caco2- | 0.5855 |
P-glycoprotein Substrate | Non-substrate | 0.7351 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9791 |
Non-inhibitor | 0.9252 |
Renal Organic Cation Transporter | Non-inhibitor | 0.8989 |
Distribution |
Subcellular localization | Mitochondria | 0.8504 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8418 |
CYP450 2D6 Substrate | Non-substrate | 0.8931 |
CYP450 3A4 Substrate | Non-substrate | 0.7786 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9088 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9043 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9707 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9622 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9543 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9759 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9462 |
Non-inhibitor | 0.9276 |
AMES Toxicity | Non AMES toxic | 0.9486 |
Carcinogens | Non-carcinogens | 0.7964 |
Fish Toxicity | Low FHMT | 0.5099 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7251 |
Honey Bee Toxicity | High HBT | 0.6594 |
Biodegradation | Ready biodegradable | 0.9364 |
Acute Oral Toxicity | III | 0.5988 |
Carcinogenicity (Three-class) | Non-required | 0.7159 |