Absorption |
Blood-Brain Barrier | BBB+ | 0.9598 |
Human Intestinal Absorption | HIA+ | 0.9186 |
Caco-2 Permeability | Caco2- | 0.5478 |
P-glycoprotein Substrate | Non-substrate | 0.9041 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9737 |
Non-inhibitor | 0.9938 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9439 |
Distribution |
Subcellular localization | Mitochondria | 0.6751 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8469 |
CYP450 2D6 Substrate | Non-substrate | 0.8370 |
CYP450 3A4 Substrate | Non-substrate | 0.7516 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8600 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8952 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9381 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8995 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9790 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9595 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.7312 |
Non-inhibitor | 0.9750 |
AMES Toxicity | Non AMES toxic | 0.8634 |
Carcinogens | Carcinogens | 0.6597 |
Fish Toxicity | Low FHMT | 0.8141 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.6467 |
Honey Bee Toxicity | High HBT | 0.7912 |
Biodegradation | Ready biodegradable | 0.8863 |
Acute Oral Toxicity | II | 0.4889 |
Carcinogenicity (Three-class) | Warning | 0.4799 |