Absorption |
Blood-Brain Barrier | BBB+ | 0.9045 |
Human Intestinal Absorption | HIA+ | 0.7927 |
Caco-2 Permeability | Caco2- | 0.7089 |
P-glycoprotein Substrate | Non-substrate | 0.8617 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9733 |
Non-inhibitor | 0.9936 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9439 |
Distribution |
Subcellular localization | Mitochondria | 0.6958 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8115 |
CYP450 2D6 Substrate | Non-substrate | 0.8472 |
CYP450 3A4 Substrate | Non-substrate | 0.7773 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9101 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9031 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9346 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9187 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9762 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9660 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.8358 |
Non-inhibitor | 0.9621 |
AMES Toxicity | Non AMES toxic | 0.8348 |
Carcinogens | Carcinogens | 0.6573 |
Fish Toxicity | Low FHMT | 0.7539 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7035 |
Honey Bee Toxicity | High HBT | 0.7409 |
Biodegradation | Not ready biodegradable | 0.6937 |
Acute Oral Toxicity | III | 0.6566 |
Carcinogenicity (Three-class) | Non-required | 0.5392 |