Absorption |
Blood-Brain Barrier | BBB+ | 0.9727 |
Human Intestinal Absorption | HIA+ | 0.7648 |
Caco-2 Permeability | Caco2+ | 0.6948 |
P-glycoprotein Substrate | Non-substrate | 0.8993 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9857 |
Non-inhibitor | 0.9857 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9265 |
Distribution |
Subcellular localization | Lysosome | 0.5251 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8261 |
CYP450 2D6 Substrate | Non-substrate | 0.7762 |
CYP450 3A4 Substrate | Non-substrate | 0.7929 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.7239 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8695 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9204 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9016 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9337 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9065 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9535 |
Non-inhibitor | 0.9680 |
AMES Toxicity | Non AMES toxic | 0.7005 |
Carcinogens | Carcinogens | 0.6865 |
Fish Toxicity | Low FHMT | 0.5387 |
Tetrahymena Pyriformis Toxicity | High TPT | 0.6557 |
Honey Bee Toxicity | High HBT | 0.8164 |
Biodegradation | Not ready biodegradable | 0.5898 |
Acute Oral Toxicity | II | 0.6940 |
Carcinogenicity (Three-class) | Non-required | 0.5624 |