Absorption |
Blood-Brain Barrier | BBB+ | 0.8653 |
Human Intestinal Absorption | HIA+ | 0.9789 |
Caco-2 Permeability | Caco2- | 0.6586 |
P-glycoprotein Substrate | Non-substrate | 0.8190 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9865 |
Non-inhibitor | 0.9915 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9496 |
Distribution |
Subcellular localization | Mitochondria | 0.7964 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8097 |
CYP450 2D6 Substrate | Non-substrate | 0.9056 |
CYP450 3A4 Substrate | Non-substrate | 0.8239 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9351 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9075 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9578 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9471 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9724 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9871 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9794 |
Non-inhibitor | 0.9826 |
AMES Toxicity | Non AMES toxic | 0.8907 |
Carcinogens | Non-carcinogens | 0.5493 |
Fish Toxicity | High FHMT | 0.7428 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9056 |
Honey Bee Toxicity | High HBT | 0.7694 |
Biodegradation | Ready biodegradable | 0.7827 |
Acute Oral Toxicity | III | 0.3902 |
Carcinogenicity (Three-class) | Non-required | 0.7092 |