Absorption |
Blood-Brain Barrier | BBB+ | 0.8705 |
Human Intestinal Absorption | HIA+ | 0.9313 |
Caco-2 Permeability | Caco2- | 0.6958 |
P-glycoprotein Substrate | Non-substrate | 0.8147 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9876 |
Non-inhibitor | 0.9911 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9524 |
Distribution |
Subcellular localization | Mitochondria | 0.7888 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8130 |
CYP450 2D6 Substrate | Non-substrate | 0.9003 |
CYP450 3A4 Substrate | Non-substrate | 0.8052 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9256 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9084 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9547 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9406 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9544 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9873 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9803 |
Non-inhibitor | 0.9844 |
AMES Toxicity | Non AMES toxic | 0.9146 |
Carcinogens | Non-carcinogens | 0.6069 |
Fish Toxicity | High FHMT | 0.7981 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9255 |
Honey Bee Toxicity | High HBT | 0.7643 |
Biodegradation | Ready biodegradable | 0.8393 |
Acute Oral Toxicity | III | 0.4559 |
Carcinogenicity (Three-class) | Non-required | 0.7340 |