Absorption |
Blood-Brain Barrier | BBB+ | 0.9661 |
Human Intestinal Absorption | HIA+ | 0.9835 |
Caco-2 Permeability | Caco2+ | 0.7599 |
P-glycoprotein Substrate | Non-substrate | 0.8904 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9847 |
Non-inhibitor | 0.9874 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9068 |
Distribution |
Subcellular localization | Lysosome | 0.7461 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8500 |
CYP450 2D6 Substrate | Non-substrate | 0.8103 |
CYP450 3A4 Substrate | Non-substrate | 0.8303 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9108 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9240 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9357 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9450 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9707 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.8311 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9391 |
Non-inhibitor | 0.9755 |
AMES Toxicity | Non AMES toxic | 0.9837 |
Carcinogens | Carcinogens | 0.6116 |
Fish Toxicity | Low FHMT | 0.5819 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8472 |
Honey Bee Toxicity | High HBT | 0.7691 |
Biodegradation | Ready biodegradable | 0.9292 |
Acute Oral Toxicity | III | 0.5994 |
Carcinogenicity (Three-class) | Non-required | 0.5999 |