Absorption |
Blood-Brain Barrier | BBB+ | 0.9852 |
Human Intestinal Absorption | HIA+ | 0.9898 |
Caco-2 Permeability | Caco2+ | 0.8078 |
P-glycoprotein Substrate | Non-substrate | 0.6792 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.8912 |
Non-inhibitor | 0.7550 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9048 |
Distribution |
Subcellular localization | Lysosome | 0.4936 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8276 |
CYP450 2D6 Substrate | Non-substrate | 0.7681 |
CYP450 3A4 Substrate | Non-substrate | 0.6822 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.6579 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9294 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9318 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9447 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9823 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.7775 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.8953 |
Non-inhibitor | 0.8127 |
AMES Toxicity | Non AMES toxic | 0.9912 |
Carcinogens | Carcinogens | 0.6985 |
Fish Toxicity | High FHMT | 0.8424 |
Tetrahymena Pyriformis Toxicity | High TPT | 0.9706 |
Honey Bee Toxicity | High HBT | 0.7799 |
Biodegradation | Ready biodegradable | 0.5915 |
Acute Oral Toxicity | IV | 0.4727 |
Carcinogenicity (Three-class) | Non-required | 0.5634 |