Absorption |
Blood-Brain Barrier | BBB+ | 0.9057 |
Human Intestinal Absorption | HIA+ | 0.9529 |
Caco-2 Permeability | Caco2- | 0.6006 |
P-glycoprotein Substrate | Non-substrate | 0.8713 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9931 |
Non-inhibitor | 0.9879 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9466 |
Distribution |
Subcellular localization | Mitochondria | 0.5978 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8393 |
CYP450 2D6 Substrate | Non-substrate | 0.9275 |
CYP450 3A4 Substrate | Non-substrate | 0.8400 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9573 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9417 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9729 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9821 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9644 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9826 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9763 |
Non-inhibitor | 0.9837 |
AMES Toxicity | Non AMES toxic | 0.9657 |
Carcinogens | Carcinogens | 0.5557 |
Fish Toxicity | Low FHMT | 0.6160 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9848 |
Honey Bee Toxicity | High HBT | 0.6666 |
Biodegradation | Ready biodegradable | 0.9659 |
Acute Oral Toxicity | III | 0.6272 |
Carcinogenicity (Three-class) | Non-required | 0.7349 |