Absorption |
Blood-Brain Barrier | BBB+ | 0.9681 |
Human Intestinal Absorption | HIA+ | 0.5891 |
Caco-2 Permeability | Caco2+ | 0.7142 |
P-glycoprotein Substrate | Non-substrate | 0.8729 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9906 |
Non-inhibitor | 0.9840 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9307 |
Distribution |
Subcellular localization | Lysosome | 0.4553 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8203 |
CYP450 2D6 Substrate | Non-substrate | 0.9073 |
CYP450 3A4 Substrate | Non-substrate | 0.8306 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8858 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9574 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9590 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9610 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9834 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9634 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9301 |
Non-inhibitor | 0.9744 |
AMES Toxicity | Non AMES toxic | 0.9015 |
Carcinogens | Carcinogens | 0.6492 |
Fish Toxicity | Low FHMT | 0.8556 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.6856 |
Honey Bee Toxicity | High HBT | 0.7868 |
Biodegradation | Ready biodegradable | 0.9026 |
Acute Oral Toxicity | II | 0.4877 |
Carcinogenicity (Three-class) | Non-required | 0.6386 |