Absorption |
Blood-Brain Barrier | BBB+ | 0.9384 |
Human Intestinal Absorption | HIA+ | 0.9419 |
Caco-2 Permeability | Caco2+ | 0.6054 |
P-glycoprotein Substrate | Non-substrate | 0.8329 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9832 |
Non-inhibitor | 0.9803 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9136 |
Distribution |
Subcellular localization | Lysosome | 0.5401 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8631 |
CYP450 2D6 Substrate | Non-substrate | 0.8156 |
CYP450 3A4 Substrate | Non-substrate | 0.8533 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9454 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8691 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9688 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9565 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9400 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.7458 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9623 |
Non-inhibitor | 0.9707 |
AMES Toxicity | Non AMES toxic | 0.9372 |
Carcinogens | Carcinogens | 0.6532 |
Fish Toxicity | Low FHMT | 0.6323 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8415 |
Honey Bee Toxicity | High HBT | 0.6508 |
Biodegradation | Ready biodegradable | 0.7024 |
Acute Oral Toxicity | II | 0.4270 |
Carcinogenicity (Three-class) | Non-required | 0.6654 |