Absorption |
Blood-Brain Barrier | BBB+ | 0.8106 |
Human Intestinal Absorption | HIA- | 0.7019 |
Caco-2 Permeability | Caco2- | 0.5645 |
P-glycoprotein Substrate | Non-substrate | 0.8165 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9881 |
Non-inhibitor | 0.9781 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9456 |
Distribution |
Subcellular localization | Mitochondria | 0.5480 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8312 |
CYP450 2D6 Substrate | Non-substrate | 0.8771 |
CYP450 3A4 Substrate | Non-substrate | 0.7862 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8757 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8775 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9401 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9047 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9447 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9515 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9611 |
Non-inhibitor | 0.9740 |
AMES Toxicity | Non AMES toxic | 0.8196 |
Carcinogens | Carcinogens | 0.5203 |
Fish Toxicity | Low FHMT | 0.9012 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9082 |
Honey Bee Toxicity | High HBT | 0.6840 |
Biodegradation | Ready biodegradable | 0.8589 |
Acute Oral Toxicity | III | 0.6050 |
Carcinogenicity (Three-class) | Non-required | 0.6653 |