Absorption |
Blood-Brain Barrier | BBB+ | 0.8218 |
Human Intestinal Absorption | HIA+ | 0.8318 |
Caco-2 Permeability | Caco2- | 0.5597 |
P-glycoprotein Substrate | Non-substrate | 0.8144 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9850 |
Non-inhibitor | 0.9791 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9421 |
Distribution |
Subcellular localization | Mitochondria | 0.5777 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8473 |
CYP450 2D6 Substrate | Non-substrate | 0.9037 |
CYP450 3A4 Substrate | Non-substrate | 0.8087 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9272 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9222 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9665 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9496 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9603 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9542 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9673 |
Non-inhibitor | 0.9792 |
AMES Toxicity | Non AMES toxic | 0.8473 |
Carcinogens | Carcinogens | 0.5590 |
Fish Toxicity | Low FHMT | 0.9076 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.9020 |
Honey Bee Toxicity | High HBT | 0.7407 |
Biodegradation | Ready biodegradable | 0.6374 |
Acute Oral Toxicity | III | 0.6084 |
Carcinogenicity (Three-class) | Non-required | 0.6720 |