Absorption |
Blood-Brain Barrier | BBB+ | 0.9453 |
Human Intestinal Absorption | HIA+ | 0.9476 |
Caco-2 Permeability | Caco2+ | 0.6166 |
P-glycoprotein Substrate | Non-substrate | 0.8495 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9757 |
Non-inhibitor | 0.9781 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9191 |
Distribution |
Subcellular localization | Lysosome | 0.4650 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8459 |
CYP450 2D6 Substrate | Non-substrate | 0.8266 |
CYP450 3A4 Substrate | Non-substrate | 0.8095 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8690 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8673 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9642 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9316 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9731 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.8425 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9572 |
Non-inhibitor | 0.9654 |
AMES Toxicity | Non AMES toxic | 0.9246 |
Carcinogens | Carcinogens | 0.6570 |
Fish Toxicity | Low FHMT | 0.6635 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7685 |
Honey Bee Toxicity | High HBT | 0.8096 |
Biodegradation | Ready biodegradable | 0.6604 |
Acute Oral Toxicity | III | 0.6171 |
Carcinogenicity (Three-class) | Non-required | 0.4958 |