Absorption |
Blood-Brain Barrier | BBB+ | 0.9203 |
Human Intestinal Absorption | HIA+ | 0.9057 |
Caco-2 Permeability | Caco2+ | 0.6082 |
P-glycoprotein Substrate | Non-substrate | 0.8451 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9888 |
Non-inhibitor | 0.9753 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9258 |
Distribution |
Subcellular localization | Lysosome | 0.6197 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8413 |
CYP450 2D6 Substrate | Non-substrate | 0.8898 |
CYP450 3A4 Substrate | Non-substrate | 0.8468 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.9322 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9140 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9601 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9525 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9706 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9032 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9306 |
Non-inhibitor | 0.9675 |
AMES Toxicity | Non AMES toxic | 0.8985 |
Carcinogens | Carcinogens | 0.6241 |
Fish Toxicity | Low FHMT | 0.8492 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8571 |
Honey Bee Toxicity | High HBT | 0.6795 |
Biodegradation | Ready biodegradable | 0.8267 |
Acute Oral Toxicity | II | 0.4615 |
Carcinogenicity (Three-class) | Non-required | 0.7416 |