Absorption |
Blood-Brain Barrier | BBB+ | 0.9354 |
Human Intestinal Absorption | HIA+ | 0.7258 |
Caco-2 Permeability | Caco2+ | 0.5655 |
P-glycoprotein Substrate | Non-substrate | 0.8706 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9838 |
Non-inhibitor | 0.9871 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9389 |
Distribution |
Subcellular localization | Mitochondria | 0.5268 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8543 |
CYP450 2D6 Substrate | Non-substrate | 0.8889 |
CYP450 3A4 Substrate | Non-substrate | 0.7916 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8913 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9239 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9533 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9355 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9619 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9380 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9438 |
Non-inhibitor | 0.9849 |
AMES Toxicity | Non AMES toxic | 0.8735 |
Carcinogens | Carcinogens | 0.5403 |
Fish Toxicity | Low FHMT | 0.8522 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8767 |
Honey Bee Toxicity | High HBT | 0.7842 |
Biodegradation | Ready biodegradable | 0.9430 |
Acute Oral Toxicity | III | 0.5882 |
Carcinogenicity (Three-class) | Non-required | 0.6246 |