Absorption |
Blood-Brain Barrier | BBB+ | 0.9750 |
Human Intestinal Absorption | HIA+ | 0.9445 |
Caco-2 Permeability | Caco2+ | 0.6764 |
P-glycoprotein Substrate | Non-substrate | 0.9039 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9891 |
Non-inhibitor | 0.9866 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9196 |
Distribution |
Subcellular localization | Lysosome | 0.4979 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8116 |
CYP450 2D6 Substrate | Non-substrate | 0.7170 |
CYP450 3A4 Substrate | Non-substrate | 0.7571 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.7506 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8586 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9306 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8304 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9560 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9002 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9433 |
Non-inhibitor | 0.9634 |
AMES Toxicity | Non AMES toxic | 0.6808 |
Carcinogens | Carcinogens | 0.7640 |
Fish Toxicity | High FHMT | 0.5199 |
Tetrahymena Pyriformis Toxicity | High TPT | 0.6171 |
Honey Bee Toxicity | High HBT | 0.8244 |
Biodegradation | Ready biodegradable | 0.6815 |
Acute Oral Toxicity | III | 0.7301 |
Carcinogenicity (Three-class) | Non-required | 0.5321 |