Absorption |
Blood-Brain Barrier | BBB+ | 0.9418 |
Human Intestinal Absorption | HIA+ | 0.9725 |
Caco-2 Permeability | Caco2+ | 0.6261 |
P-glycoprotein Substrate | Non-substrate | 0.8455 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9786 |
Non-inhibitor | 0.9781 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9142 |
Distribution |
Subcellular localization | Lysosome | 0.5526 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8473 |
CYP450 2D6 Substrate | Non-substrate | 0.8257 |
CYP450 3A4 Substrate | Non-substrate | 0.8090 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8748 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8802 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9691 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9372 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9832 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.8287 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9621 |
Non-inhibitor | 0.9639 |
AMES Toxicity | Non AMES toxic | 0.9194 |
Carcinogens | Carcinogens | 0.6655 |
Fish Toxicity | Low FHMT | 0.6285 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7685 |
Honey Bee Toxicity | High HBT | 0.7757 |
Biodegradation | Ready biodegradable | 0.5241 |
Acute Oral Toxicity | III | 0.5606 |
Carcinogenicity (Three-class) | Non-required | 0.5025 |