Absorption |
Blood-Brain Barrier | BBB+ | 0.9455 |
Human Intestinal Absorption | HIA+ | 0.9726 |
Caco-2 Permeability | Caco2+ | 0.6509 |
P-glycoprotein Substrate | Non-substrate | 0.8460 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9807 |
Non-inhibitor | 0.9784 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9145 |
Distribution |
Subcellular localization | Lysosome | 0.5561 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8620 |
CYP450 2D6 Substrate | Non-substrate | 0.8297 |
CYP450 3A4 Substrate | Non-substrate | 0.8176 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8963 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8848 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9744 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9506 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9862 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.8225 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9621 |
Non-inhibitor | 0.9663 |
AMES Toxicity | Non AMES toxic | 0.9390 |
Carcinogens | Carcinogens | 0.6791 |
Fish Toxicity | Low FHMT | 0.6292 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.7918 |
Honey Bee Toxicity | High HBT | 0.7830 |
Biodegradation | Not ready biodegradable | 0.5239 |
Acute Oral Toxicity | III | 0.5553 |
Carcinogenicity (Three-class) | Non-required | 0.4947 |