Absorption |
Blood-Brain Barrier | BBB+ | 0.9771 |
Human Intestinal Absorption | HIA+ | 0.9929 |
Caco-2 Permeability | Caco2+ | 0.7249 |
P-glycoprotein Substrate | Non-substrate | 0.8972 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9778 |
Non-inhibitor | 0.9790 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9103 |
Distribution |
Subcellular localization | Lysosome | 0.6313 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8422 |
CYP450 2D6 Substrate | Non-substrate | 0.6657 |
CYP450 3A4 Substrate | Non-substrate | 0.7960 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.7671 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8619 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9629 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8947 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9667 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.8858 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9688 |
Non-inhibitor | 0.9675 |
AMES Toxicity | AMES toxic | 0.7931 |
Carcinogens | Carcinogens | 0.7287 |
Fish Toxicity | Low FHMT | 0.5210 |
Tetrahymena Pyriformis Toxicity | High TPT | 0.9712 |
Honey Bee Toxicity | High HBT | 0.8421 |
Biodegradation | Not ready biodegradable | 0.7008 |
Acute Oral Toxicity | II | 0.4938 |
Carcinogenicity (Three-class) | Warning | 0.5391 |