Absorption |
Blood-Brain Barrier | BBB+ | 0.9839 |
Human Intestinal Absorption | HIA+ | 0.9951 |
Caco-2 Permeability | Caco2+ | 0.7367 |
P-glycoprotein Substrate | Non-substrate | 0.8941 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9667 |
Non-inhibitor | 0.9817 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9208 |
Distribution |
Subcellular localization | Lysosome | 0.5125 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8433 |
CYP450 2D6 Substrate | Non-substrate | 0.7372 |
CYP450 3A4 Substrate | Non-substrate | 0.8004 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.7842 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9128 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9632 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9306 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9719 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9115 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9713 |
Non-inhibitor | 0.9598 |
AMES Toxicity | Non AMES toxic | 0.8490 |
Carcinogens | Carcinogens | 0.7612 |
Fish Toxicity | Low FHMT | 0.5943 |
Tetrahymena Pyriformis Toxicity | High TPT | 0.7847 |
Honey Bee Toxicity | High HBT | 0.8319 |
Biodegradation | Not ready biodegradable | 0.8276 |
Acute Oral Toxicity | III | 0.6906 |
Carcinogenicity (Three-class) | Warning | 0.4752 |