Absorption |
Blood-Brain Barrier | BBB+ | 0.9624 |
Human Intestinal Absorption | HIA+ | 0.9436 |
Caco-2 Permeability | Caco2+ | 0.6505 |
P-glycoprotein Substrate | Non-substrate | 0.8690 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9785 |
Non-inhibitor | 0.9835 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9239 |
Distribution |
Subcellular localization | Lysosome | 0.4689 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8203 |
CYP450 2D6 Substrate | Non-substrate | 0.8890 |
CYP450 3A4 Substrate | Non-substrate | 0.8149 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.7991 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9121 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9416 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9066 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9734 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9461 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9380 |
Non-inhibitor | 0.9706 |
AMES Toxicity | Non AMES toxic | 0.7897 |
Carcinogens | Carcinogens | 0.6445 |
Fish Toxicity | Low FHMT | 0.8625 |
Tetrahymena Pyriformis Toxicity | High TPT | 0.5378 |
Honey Bee Toxicity | High HBT | 0.7814 |
Biodegradation | Ready biodegradable | 0.7239 |
Acute Oral Toxicity | II | 0.4302 |
Carcinogenicity (Three-class) | Non-required | 0.6219 |