Absorption |
Blood-Brain Barrier | BBB+ | 0.9725 |
Human Intestinal Absorption | HIA+ | 0.9687 |
Caco-2 Permeability | Caco2+ | 0.6957 |
P-glycoprotein Substrate | Non-substrate | 0.8877 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9732 |
Non-inhibitor | 0.9855 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9154 |
Distribution |
Subcellular localization | Lysosome | 0.4862 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8289 |
CYP450 2D6 Substrate | Non-substrate | 0.8233 |
CYP450 3A4 Substrate | Non-substrate | 0.8075 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8726 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.9266 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9657 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.9452 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9803 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.8881 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.9489 |
Non-inhibitor | 0.9737 |
AMES Toxicity | Non AMES toxic | 0.9503 |
Carcinogens | Carcinogens | 0.6480 |
Fish Toxicity | Low FHMT | 0.6535 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.6398 |
Honey Bee Toxicity | High HBT | 0.8474 |
Biodegradation | Ready biodegradable | 0.8278 |
Acute Oral Toxicity | III | 0.6385 |
Carcinogenicity (Three-class) | Non-required | 0.4650 |