Absorption |
Blood-Brain Barrier | BBB+ | 0.9321 |
Human Intestinal Absorption | HIA- | 0.5000 |
Caco-2 Permeability | Caco2- | 0.6797 |
P-glycoprotein Substrate | Non-substrate | 0.8763 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9321 |
Non-inhibitor | 0.9919 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9528 |
Distribution |
Subcellular localization | Mitochondria | 0.5454 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8323 |
CYP450 2D6 Substrate | Non-substrate | 0.8247 |
CYP450 3A4 Substrate | Non-substrate | 0.7299 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8642 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8410 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9137 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8559 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9867 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9814 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.8806 |
Non-inhibitor | 0.9240 |
AMES Toxicity | Non AMES toxic | 0.8908 |
Carcinogens | Carcinogens | 0.8269 |
Fish Toxicity | Low FHMT | 0.5560 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8210 |
Honey Bee Toxicity | High HBT | 0.7265 |
Biodegradation | Not ready biodegradable | 0.5830 |
Acute Oral Toxicity | III | 0.7594 |
Carcinogenicity (Three-class) | Non-required | 0.7075 |