Absorption |
Blood-Brain Barrier | BBB+ | 0.9359 |
Human Intestinal Absorption | HIA- | 0.5000 |
Caco-2 Permeability | Caco2- | 0.6921 |
P-glycoprotein Substrate | Non-substrate | 0.8768 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9362 |
Non-inhibitor | 0.9920 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9532 |
Distribution |
Subcellular localization | Mitochondria | 0.5505 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8323 |
CYP450 2D6 Substrate | Non-substrate | 0.8280 |
CYP450 3A4 Substrate | Non-substrate | 0.7365 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8890 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8605 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9232 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8812 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9901 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9832 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.8806 |
Non-inhibitor | 0.9272 |
AMES Toxicity | Non AMES toxic | 0.9132 |
Carcinogens | Carcinogens | 0.8357 |
Fish Toxicity | Low FHMT | 0.5566 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8415 |
Honey Bee Toxicity | High HBT | 0.7369 |
Biodegradation | Not ready biodegradable | 0.5815 |
Acute Oral Toxicity | III | 0.7802 |
Carcinogenicity (Three-class) | Non-required | 0.7149 |