Absorption |
Blood-Brain Barrier | BBB+ | 0.9336 |
Human Intestinal Absorption | HIA+ | 0.6352 |
Caco-2 Permeability | Caco2- | 0.6851 |
P-glycoprotein Substrate | Non-substrate | 0.8374 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9305 |
Non-inhibitor | 0.9923 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9555 |
Distribution |
Subcellular localization | Mitochondria | 0.5541 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.7771 |
CYP450 2D6 Substrate | Non-substrate | 0.8318 |
CYP450 3A4 Substrate | Non-substrate | 0.7208 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8850 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.8647 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9222 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8828 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9899 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9834 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.8646 |
Non-inhibitor | 0.9231 |
AMES Toxicity | Non AMES toxic | 0.9056 |
Carcinogens | Carcinogens | 0.8578 |
Fish Toxicity | Low FHMT | 0.5441 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8472 |
Honey Bee Toxicity | High HBT | 0.7223 |
Biodegradation | Not ready biodegradable | 0.7138 |
Acute Oral Toxicity | III | 0.7544 |
Carcinogenicity (Three-class) | Non-required | 0.7035 |