Absorption |
Blood-Brain Barrier | BBB+ | 0.9312 |
Human Intestinal Absorption | HIA- | 0.6825 |
Caco-2 Permeability | Caco2- | 0.6544 |
P-glycoprotein Substrate | Non-substrate | 0.8777 |
P-glycoprotein Inhibitor | Non-inhibitor | 0.9450 |
Non-inhibitor | 0.9870 |
Renal Organic Cation Transporter | Non-inhibitor | 0.9581 |
Distribution |
Subcellular localization | Mitochondria | 0.5495 |
Metabolism |
CYP450 2C9 Substrate | Non-substrate | 0.8713 |
CYP450 2D6 Substrate | Non-substrate | 0.8206 |
CYP450 3A4 Substrate | Non-substrate | 0.7189 |
CYP450 1A2 Inhibitor | Non-inhibitor | 0.8299 |
CYP450 2C9 Inhibitor | Non-inhibitor | 0.7930 |
CYP450 2D6 Inhibitor | Non-inhibitor | 0.9154 |
CYP450 2C19 Inhibitor | Non-inhibitor | 0.8183 |
CYP450 3A4 Inhibitor | Non-inhibitor | 0.9865 |
CYP Inhibitory Promiscuity | Low CYP Inhibitory Promiscuity | 0.9784 |
Excretion |
Toxicity |
Human Ether-a-go-go-Related Gene Inhibition | Weak inhibitor | 0.8522 |
Non-inhibitor | 0.9262 |
AMES Toxicity | Non AMES toxic | 0.7718 |
Carcinogens | Carcinogens | 0.8220 |
Fish Toxicity | Low FHMT | 0.7382 |
Tetrahymena Pyriformis Toxicity | Low TPT | 0.8466 |
Honey Bee Toxicity | High HBT | 0.7245 |
Biodegradation | Ready biodegradable | 0.8064 |
Acute Oral Toxicity | III | 0.6693 |
Carcinogenicity (Three-class) | Non-required | 0.6904 |