General Information

MaintermPOLYPROPYLENE GLYCOL (M W 1,200-3,000)
Doc TypeASP
CAS Reg.No.(or other ID)25322-69-4
Regnum 175.105
175.300
177.1680
178.3740
173.310
173.340

From www.fda.gov

Computed Descriptors

Download SDF
2D Structure
CID32881
IUPAC Name2-(2-hydroxypropoxy)propan-1-ol
InChIInChI=1S/C6H14O3/c1-5(8)4-9-6(2)3-7/h5-8H,3-4H2,1-2H3
InChI KeyDUFKCOQISQKSAV-UHFFFAOYSA-N
Canonical SMILESCC(CO)OCC(C)O
Molecular FormulaC6H14O3
Wikipedia2-(2-hydroxypropoxy)propan-1-ol

From Pubchem


Computed Properties

Property Name Property Value
Molecular Weight134.175
Hydrogen Bond Donor Count2
Hydrogen Bond Acceptor Count3
Rotatable Bond Count4
Complexity65.3
CACTVS Substructure Key Fingerprint A A A D c c B g M A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A G g A A C A A A C B S g g A I C A A A A B g A A A A A A A A A A A A A A A A A A A A A A A A A B E A A A A A A C Q A A A A A A D A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A = =
Topological Polar Surface Area49.7
Monoisotopic Mass134.094
Exact Mass134.094
Compound Is CanonicalizedTrue
Formal Charge0
Heavy Atom Count9
Defined Atom Stereocenter Count0
Undefined Atom Stereocenter Count2
Defined Bond Stereocenter Count0
Undefined Bond Stereocenter Count0
Isotope Atom Count0
Covalently-Bonded Unit Count1

From Pubchem


ADMET Predicted Profile --- Classification

Model Result Probability
Absorption
Blood-Brain BarrierBBB+0.8060
Human Intestinal AbsorptionHIA+0.9697
Caco-2 PermeabilityCaco2-0.5218
P-glycoprotein SubstrateSubstrate0.5259
P-glycoprotein InhibitorNon-inhibitor0.8368
Non-inhibitor0.7466
Renal Organic Cation TransporterNon-inhibitor0.8985
Distribution
Subcellular localizationMitochondria0.7175
Metabolism
CYP450 2C9 SubstrateNon-substrate0.8332
CYP450 2D6 SubstrateNon-substrate0.8388
CYP450 3A4 SubstrateNon-substrate0.6895
CYP450 1A2 InhibitorNon-inhibitor0.8585
CYP450 2C9 InhibitorNon-inhibitor0.9003
CYP450 2D6 InhibitorNon-inhibitor0.9152
CYP450 2C19 InhibitorNon-inhibitor0.8284
CYP450 3A4 InhibitorNon-inhibitor0.9289
CYP Inhibitory PromiscuityLow CYP Inhibitory Promiscuity0.9051
Excretion
Toxicity
Human Ether-a-go-go-Related Gene InhibitionWeak inhibitor0.9731
Non-inhibitor0.7661
AMES ToxicityNon AMES toxic0.8097
CarcinogensCarcinogens 0.5256
Fish ToxicityLow FHMT0.6829
Tetrahymena Pyriformis ToxicityLow TPT0.9853
Honey Bee ToxicityHigh HBT0.6869
BiodegradationNot ready biodegradable0.6859
Acute Oral ToxicityIII0.5927
Carcinogenicity (Three-class)Non-required0.7608

From admetSAR


ADMET Predicted Profile --- Regression

Model Value Unit
Absorption
Aqueous solubility-0.0537LogS
Caco-2 Permeability0.7225LogPapp, cm/s
Distribution
Metabolism
Excretion
Toxicity
Rat Acute Toxicity1.2940LD50, mol/kg
Fish Toxicity3.7305pLC50, mg/L
Tetrahymena Pyriformis Toxicity-1.6612pIGC50, ug/L

From admetSAR


Toxicity Profile

Route of Exposure
Mechanism of Toxicity
Metabolism
Toxicity Values
Lethal Dose
Carcinogenicity (IARC Classification)No indication of carcinogenicity to humans (not listed by IARC).
Minimum Risk Level
Health Effects
Treatment
Reference

From T3DB


Taxonomic Classification

KingdomOrganic compounds
SuperclassOrganic oxygen compounds
ClassOrganooxygen compounds
SubclassAlcohols and polyols
Intermediate Tree NodesNot available
Direct ParentSecondary alcohols
Alternative Parents
Molecular FrameworkAliphatic acyclic compounds
SubstituentsSecondary alcohol - Ether - Dialkyl ether - Hydrocarbon derivative - Primary alcohol - Aliphatic acyclic compound
DescriptionThis compound belongs to the class of organic compounds known as secondary alcohols. These are compounds containing a secondary alcohol functional group, with the general structure HOC(R)(R') (R,R'=alkyl, aryl).

From ClassyFire


Targets

General Function:
Zinc ion binding
Specific Function:
Orphan receptor that acts as transcription activator in the absence of bound ligand. Binds specifically to an estrogen response element and activates reporter genes controlled by estrogen response elements (By similarity). Induces the expression of PERM1 in the skeletal muscle.
Gene Name:
ESRRG
Uniprot ID:
P62508
Molecular Weight:
51305.485 Da
References
  1. Sipes NS, Martin MT, Kothiya P, Reif DM, Judson RS, Richard AM, Houck KA, Dix DJ, Kavlock RJ, Knudsen TB: Profiling 976 ToxCast chemicals across 331 enzymatic and receptor signaling assays. Chem Res Toxicol. 2013 Jun 17;26(6):878-95. doi: 10.1021/tx400021f. Epub 2013 May 16. [23611293 ]

From T3DB