General Information

Chemical Names: CITRANAXANTHIN; 6'-METHYL-6'-apo-beta-CAROTEN-6'-ONE; 5',6'-DEHYDRO-5'-apo-18'-NOR-beta-CAROTEN-6'-ONE
CAS number: 3604-90-8
Functional Class: Food Additives
COLOUR

From apps.who.int


Evaluations

Evaluation year: 1987
ADI: NO ADI ALLOCATED
Meeting: 31
Specs Code: R
Report: TRS 759-JECFA 31/27
Tox Monograph: FAS 22-JECFA 31/85
Specification: COMPENDIUM ADDENDUM 12/FNP 52 Add. 12/67 (METALS LIMITS) (2004); FAO JECFA Monographs 1 vol.1/397

From apps.who.int


Computed Descriptors

Download SDF
2D Structure
CID6436724
IUPAC Name(3E,5E,7E,9E,11E,13E,15E,17E,19E)-5,9,14,18-tetramethyl-20-(2,6,6-trimethylcyclohexen-1-yl)icosa-3,5,7,9,11,13,15,17,19-nonaen-2-one
InChIInChI=1S/C33H44O/c1-26(16-11-18-28(3)21-23-31(6)34)14-9-10-15-27(2)17-12-19-29(4)22-24-32-30(5)20-13-25-33(32,7)8/h9-12,14-19,21-24H,13,20,25H2,1-8H3/b10-9+,16-11+,17-12+,23-21+,24-22+,26-14+,27-15+,28-18+,29-19+
InChI KeyPRDJTOVRIHGKNU-ZWERVMMHSA-N
Canonical SMILESCC1=C(C(CCC1)(C)C)C=CC(=CC=CC(=CC=CC=C(C)C=CC=C(C)C=CC(=O)C)C)C
Molecular FormulaC33H44O
Wikipediacitranaxanthin

From Pubchem


Computed Properties

Property Name Property Value
Molecular Weight456.714
Hydrogen Bond Donor Count0
Hydrogen Bond Acceptor Count1
Rotatable Bond Count10
Complexity1000.0
CACTVS Substructure Key Fingerprint A A A D c f B 8 I A A A A A A A A A A A A A A A A A A A A A A A A A A g A A A A A A A A A A A A A A A A G g A A A A A A D g S A g A A C A A A A A A C I A q B S A A A A A A A g A A A I C A A A A E g I A A I A A Q A A A A A A g A A I g Y M A g M A P A A A A A A A A A A A A A A A A A A A A A A A A A A A A A A = =
Topological Polar Surface Area17.1
Monoisotopic Mass456.339
Exact Mass456.339
Compound Is CanonicalizedTrue
Formal Charge0
Heavy Atom Count34
Defined Atom Stereocenter Count0
Undefined Atom Stereocenter Count0
Defined Bond Stereocenter Count9
Undefined Bond Stereocenter Count0
Isotope Atom Count0
Covalently-Bonded Unit Count1

From Pubchem


ADMET Predicted Profile --- Classification

Model Result Probability
Absorption
Blood-Brain BarrierBBB+0.9667
Human Intestinal AbsorptionHIA+1.0000
Caco-2 PermeabilityCaco2+0.7833
P-glycoprotein SubstrateNon-substrate0.5587
P-glycoprotein InhibitorNon-inhibitor0.5853
Non-inhibitor0.5401
Renal Organic Cation TransporterNon-inhibitor0.7848
Distribution
Subcellular localizationLysosome0.4058
Metabolism
CYP450 2C9 SubstrateNon-substrate0.8506
CYP450 2D6 SubstrateNon-substrate0.8609
CYP450 3A4 SubstrateSubstrate0.6196
CYP450 1A2 InhibitorNon-inhibitor0.7697
CYP450 2C9 InhibitorNon-inhibitor0.8616
CYP450 2D6 InhibitorNon-inhibitor0.9513
CYP450 2C19 InhibitorNon-inhibitor0.8316
CYP450 3A4 InhibitorNon-inhibitor0.9491
CYP Inhibitory PromiscuityLow CYP Inhibitory Promiscuity0.6895
Excretion
Toxicity
Human Ether-a-go-go-Related Gene InhibitionWeak inhibitor0.8862
Non-inhibitor0.8869
AMES ToxicityNon AMES toxic0.9132
CarcinogensNon-carcinogens0.6926
Fish ToxicityHigh FHMT0.8766
Tetrahymena Pyriformis ToxicityHigh TPT0.8403
Honey Bee ToxicityHigh HBT0.8298
BiodegradationReady biodegradable0.6605
Acute Oral ToxicityIII0.7883
Carcinogenicity (Three-class)Non-required0.5366

From admetSAR


ADMET Predicted Profile --- Regression

Model Value Unit
Absorption
Aqueous solubility-2.2407LogS
Caco-2 Permeability1.9848LogPapp, cm/s
Distribution
Metabolism
Excretion
Toxicity
Rat Acute Toxicity1.6532LD50, mol/kg
Fish Toxicity0.5815pLC50, mg/L
Tetrahymena Pyriformis Toxicity0.1648pIGC50, ug/L

From admetSAR


Taxonomic Classification

KingdomOrganic compounds
SuperclassLipids and lipid-like molecules
ClassPrenol lipids
SubclassTriterpenoids
Intermediate Tree NodesNot available
Direct ParentTriterpenoids
Alternative Parents
Molecular FrameworkAliphatic homomonocyclic compounds
SubstituentsTriterpenoid - Alpha,beta-unsaturated ketone - Enone - Acryloyl-group - Ketone - Organic oxygen compound - Organic oxide - Hydrocarbon derivative - Organooxygen compound - Carbonyl group - Aliphatic homomonocyclic compound
DescriptionThis compound belongs to the class of organic compounds known as triterpenoids. These are terpene molecules containing six isoprene units.

From ClassyFire